Reaction Details Report a problem with these data
Target
Protease
Ligand
BDBM50163737
Substrate
n/a
Meas. Tech.
ChEMBL_1576370 (CHEMBL3802587)
IC50
6.0±n/a nM
Citation
Zhan, P; Pannecouque, C; De Clercq, E; Liu, X Anti-HIV Drug Discovery and Development: Current Innovations and Future Trends. J Med Chem 59:2849-78 (2016) [PubMed] Article
More Info.:
Target
Name:
Protease
Synonyms:
n/a
Type:
Enzyme
Mol. Mass.:
10904.79
Organism:
Human immunodeficiency virus 1 (HIV-1)
Description:
Q9YQ12
Residue:
99
Sequence:
PQITLWQRPFVTIKIEGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQIVIEICGKKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF