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Target
C-terminal-binding protein 2
Ligand
BDBM50304072
Substrate
n/a
Meas. Tech.
ChEMBL_1574551 (CHEMBL3804623)
IC50
>300000±n/a nM
Citation
 Korwar, S; Morris, BL; Parikh, HI; Coover, RA; Doughty, TW; Love, IM; Hilbert, BJ; Royer, WE; Kellogg, GE; Grossman, SR; Ellis, KC Design, synthesis, and biological evaluation of substrate-competitive inhibitors of C-terminal Binding Protein (CtBP). Bioorg Med Chem 24:2707-15 (2016) [PubMed]  Article 
Target
Name:
C-terminal-binding protein 2
Synonyms:
C-terminal-binding protein 2 | C-terminal-binding protein 2 (CtBP2) | CTBP2 | CTBP2_HUMAN
Type:
Protein
Mol. Mass.:
48948.33
Organism:
Homo sapiens (Human)
Description:
P56545
Residue:
445
Sequence:
MALVDKHKVKRQRLDRICEGIRPQIMNGPLHPRPLVALLDGRDCTVEMPILKDLATVAFCDAQSTQEIHEKVLNEAVGAMMYHTITLTREDLEKFKALRVIVRIGSGYDNVDIKAAGELGIAVCNIPSAAVEETADSTICHILNLYRRNTWLYQALREGTRVQSVEQIREVASGAARIRGETLGLIGFGRTGQAVAVRAKAFGFSVIFYDPYLQDGIERSLGVQRVYTLQDLLYQSDCVSLHCNLNEHNHHLINDFTIKQMRQGAFLVNAARGGLVDEKALAQALKEGRIRGAALDVHESEPFSFAQGPLKDAPNLICTPHTAWYSEQASLEMREAAATEIRRAITGRIPESLRNCVNKEFFVTSAPWSVIDQQAIHPELNGATYRYPPGIVGVAPGGLPAAMEGIIPGGIPVTHNLPTVAHPSQAPSPNQPTKHGDNREHPNEQ
  
Inhibitor
Name:
BDBM50304072
Synonyms:
3-PHENYLPROPIONIC ACID3-Phenyl-propionic acid | 3-phenylpropanoic acid | CHEMBL851 | HYDROCINNAMIC ACID | Phenyl propionic acid
Type:
Small organic molecule
Emp. Form.:
C9H10O2
Mol. Mass.:
150.1745
SMILES:
OC(=O)CCc1ccccc1
Structure:
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