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Target
Free fatty acid receptor 1
Ligand
BDBM50425662
Substrate
n/a
Meas. Tech.
ChEMBL_1585168 (CHEMBL3820976)
Ki
204±n/a nM
Citation
 Christiansen, E; Hudson, BD; Hansen, AH; Milligan, G; Ulven, T Development and Characterization of a Potent Free Fatty Acid Receptor 1 (FFA1) Fluorescent Tracer. J Med Chem 59:4849-58 (2016) [PubMed]  Article 
Target
Name:
Free fatty acid receptor 1
Synonyms:
FFAR1 | FFAR1_HUMAN | G-protein Coupled Receptor 40 | GPR40
Type:
G Protein-Coupled Receptor (GPCR)
Mol. Mass.:
31473.32
Organism:
Homo sapiens (Human)
Description:
O14842
Residue:
300
Sequence:
MDLPPQLSFGLYVAAFALGFPLNVLAIRGATAHARLRLTPSLVYALNLGCSDLLLTVSLPLKAVEALASGAWPLPASLCPVFAVAHFFPLYAGGGFLAALSAGRYLGAAFPLGYQAFRRPCYSWGVCAAIWALVLCHLGLVFGLEAPGGWLDHSNTSLGINTPVNGSPVCLEAWDPASAGPARFSLSLLLFFLPLAITAFCYVGCLRALARSGLTHRRKLRAAWVAGGALLTLLLCVGPYNASNVASFLYPNLGGSWRKLGLITGAWSVVLNPLVTGYLGRGPGLKTVCAARTQGGKSQK
  
Inhibitor
Name:
BDBM50425662
Synonyms:
CHEMBL2315528
Type:
Small organic molecule
Emp. Form.:
C19H15NO2
Mol. Mass.:
289.3279
SMILES:
OC(=O)CCc1ccc(cc1)C#Cc1ccccc1CC#N
Structure:
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