Reaction Details Report a problem with these data
Target
Free fatty acid receptor 4
Ligand
BDBM50196402
Substrate
n/a
Meas. Tech.
ChEMBL_1618437 (CHEMBL3860606)
EC50
72±n/a nM
Citation
 Azevedo, CM; Watterson, KR; Wargent, ET; Hansen, SV; Hudson, BD; Kepczynska, MA; Dunlop, J; Shimpukade, B; Christiansen, E; Milligan, G; Stocker, CJ; Ulven, T Non-Acidic Free Fatty Acid Receptor 4 Agonists with Antidiabetic Activity. J Med Chem 59:8868-8878 (2016) [PubMed]  Article 
Target
Name:
Free fatty acid receptor 4
Synonyms:
FFAR4_MOUSE | Ffar4 | Free fatty acid receptor 4 | G-protein coupled receptor GT01 | Gpr120 | O3far1 | Omega-3 fatty acid receptor 1
Type:
PROTEIN
Mol. Mass.:
40828.60
Organism:
Mus musculus
Description:
ChEMBL_1454435
Residue:
361
Sequence:
MSPECAQTTGPGPSHTLDQVNRTHFPFFSDVKGDHRLVLSVVETTVLGLIFVVSLLGNVCALVLVARRRRRGATASLVLNLFCADLLFTSAIPLVLVVRWTEAWLLGPVVCHLLFYVMTMSGSVTILTLAAVSLERMVCIVRLRRGLSGPGRRTQAALLAFIWGYSALAALPLCILFRVVPQRLPGGDQEIPICTLDWPNRIGEISWDVFFVTLNFLVPGLVIVISYSKILQITKASRKRLTLSLAYSESHQIRVSQQDYRLFRTLFLLMVSFFIMWSPIIITILLILIQNFRQDLVIWPSLFFWVVAFTFANSALNPILYNMSLFRNEWRKIFCCFFFPEKGAIFTDTSVRRNDLSVISS
  
Inhibitor
Name:
BDBM50196402
Synonyms:
CHEMBL3910333
Type:
Small organic molecule
Emp. Form.:
C18H13ClN2O3S
Mol. Mass.:
372.825
SMILES:
Clc1cc(Oc2ccccn2)cc(c1)N1Cc2ccccc2S1(=O)=O
Structure:
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