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Target
Free fatty acid receptor 1
Ligand
BDBM50232522
Substrate
n/a
Meas. Tech.
ChEBML_1647940
EC50
6213±n/a nM
Citation
Sparks, SM; Aquino, C; Banker, P; Collins, JL; Cowan, D; Diaz, C; Dock, ST; Hertzog, DL; Liang, X; Swiger, ED; Yuen, J; Chen, G; Jayawickreme, C; Moncol, D; Nystrom, C; Rash, V; Rimele, T; Roller, S; Ross, S Exploration of phenylpropanoic acids as agonists of the free fatty acid receptor 4 (FFA4): Identification of an orally efficacious FFA4 agonist. Bioorg Med Chem Lett 27:1278-1283 (2017) [PubMed] Article
More Info.:
Target
Name:
Free fatty acid receptor 1
Synonyms:
FFAR1_MOUSE | Ffar1 | Gpr40
Type:
PROTEIN
Mol. Mass.:
31818.80
Organism:
Mus musculus
Description:
ChEMBL_1454431
Residue:
300
Sequence:
MDLPPQLSFALYVSAFALGFPLNLLAIRGAVSHAKLRLTPSLVYTLHLGCSDLLLAITLPLKAVEALASGAWPLPLPFCPVFALAHFAPLYAGGGFLAALSAGRYLGAAFPFGYQAIRRPRYSWGVCVAIWALVLCHLGLALGLETSGSWLDNSTSSLGINIPVNGSPVCLEAWDPDSARPARLSFSILLFFLPLVITAFCYVGCLRALVRSGLSHKRKLRAAWVAGGALLTLLLCLGPYNASNVASFINPDLGGSWRKLGLITGAWSVVLNPLVTGYLGTGPGRGTICVTRTQRGTIQK