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Target
Interleukin-15
Ligand
BDBM50238643
Substrate
n/a
Meas. Tech.
ChEMBL_1664049 (CHEMBL4013730)
Kd
26000±n/a nM
Citation
Quéméner, A; Maillasson, M; Arzel, L; Sicard, B; Vomiandry, R; Mortier, E; Dubreuil, D; Jacques, Y; Lebreton, J; Mathé-Allainmat, M Discovery of a Small-Molecule Inhibitor of Interleukin 15: Pharmacophore-Based Virtual Screening and Hit Optimization. J Med Chem 60:6249-6272 (2017) [PubMed] Article
More Info.:
Target
Name:
Interleukin-15
Synonyms:
IL-15 | IL15 | IL15-IL15 receptor | IL15_HUMAN | Interleukin-15
Type:
PROTEIN
Mol. Mass.:
18080.13
Organism:
Homo sapiens
Description:
ChEMBL_117698
Residue:
162
Sequence:
MRISKPHLRSISIQCYLCLLLNSHFLTEAGIHVFILGCFSAGLPKTEANWVNVISDLKKIEDLIQSMHIDATLYTESDVHPSCKVTAMKCFLLELQVISLESGDASIHDTVENLIILANNSLSSNGNVTESGCKECEELEEKNIKEFLQSFVHIVQMFINTS