Reaction Details
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Somatostatin receptor type 3
Ligand
BDBM84944
Substrate
n/a
Ki
1000±n/a nM
Comments
PDSP_3361
Citation
Reisine, T; Bell, GI Molecular biology of somatostatin receptors. Endocr Rev 16:427-42 (1995) [PubMed] Article More Info.:
Target
Name:
Somatostatin receptor type 3
Synonyms:
SOMATOSTATIN SST3 | SS-3-R | SS3-R | SS3R | SSR-28 | SSR3_HUMAN | SSTR3 | Somatostatin receptor type 3 (SSTR3)
Type:
Protein
Mol. Mass.:
45855.97
Organism:
Homo sapiens (Human)
Description:
P32745
Residue:
418
Sequence:
MDMLHPSSVSTTSEPENASSAWPPDATLGNVSAGPSPAGLAVSGVLIPLVYLVVCVVGLLGNSLVIYVVLRHTASPSVTNVYILNLALADELFMLGLPFLAAQNALSYWPFGSLMCRLVMAVDGINQFTSIFCLTVMSVDRYLAVVHPTRSARWRTAPVARTVSAAVWVASAVVVLPVVVFSGVPRGMSTCHMQWPEPAAAWRAGFIIYTAALGFFGPLLVICLCYLLIVVKVRSAGRRVWAPSCQRRRRSERRVTRMVVAVVALFVLCWMPFYVLNIVNVVCPLPEEPAFFGLYFLVVALPYANSCANPILYGFLSYRFKQGFRRVLLRPSRRVRSQEPTVGPPEKTEEEDEEEEDGEESREGGKGKEMNGRVSQITQPGTSGQERPPSRVASKEQQLLPQEASTGEKSSTMRISYL
Inhibitor
Name:
BDBM84944
Synonyms:
cyclo[Ahep-Phe-DTrp-Lys-Thr(Bzl)]
Type:
Small organic molecule
Emp. Form.:
C43H59N7O5
Mol. Mass.:
753.9725
SMILES:
C[C@@H](Oc1ccccc1)[C@@H]1NC(O)[C@H](CCCCN)NC(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](Cc2ccccc2)NCCCCCCCNC1=O
Structure:
