Target
Neuropeptide Y receptor type 5
Ligand
BDBM82287
Substrate
n/a
Ki
8.9±n/a nM
Comments
PDSP_1387
Citation
 Weinberg, DHSirinathsinghji, DJTan, CPShiao, LLMorin, NRigby, MRHeavens, RHRapoport, DRBayne, MLCascieri, MAStrader, CDLinemeyer, DLMacNeil, DJ Cloning and expression of a novel neuropeptide Y receptor. J Biol Chem 271:16435-8 (1996) [PubMed]  Article 
Target
Name:
Neuropeptide Y receptor type 5
Synonyms:
NPY-Y5 | NPY5R_MOUSE | Neuropeptide Y receptor Y5 | Neuropeptide Y receptor type 5 (NPY Y5) | Npy5 | Npy5r
Type:
Enzyme
Mol. Mass.:
52807.91
Organism:
Mus musculus (Mouse)
Description:
O70342
Residue:
466
Sequence:
MEVKLEEHFNKTFVTENNTAASQNTASPAWEDYRGTENNTSAARNTAFPVWEDYRGSVDDLQYFLIGLYTFVSLLGFMGNLLILMAVMKKRNQKTTVNFLIGNLAFSDILVVLFCSPFTLTSVLLDQWMFGKAMCHIMPFLQCVSVLVSTLILISIAIVRYHMIKHPISNNLTANHGYFLIATVWTLGFAICSPLPVFHSLVELKETFGSALLSSKYLCVESWPSDSYRIAFTISLLLVQYILPLVCLTVSHTSVCRSISCGLSHKENRLEENEMINLTLHPSKKSRDQAKPPSTQKWSYSFIRKHRRRYSKKTACVLPAPAGPSQEKHLTVPENPGSVRSQLSPSSKVIPGVPICFEVKPEESSDAQEMRVKRSLTRIKKRSRSVFYRLTILILVFAVSWMPLHVFHVVTDFNDNLISNRHFKLVYCICHLLGMMSCCLNPILYGFLNNGIKADLRALIHCLHMS
  
Inhibitor
Name:
BDBM82287
Synonyms:
NPY2-36 | NPY2-36, human | NPY2-36, porcine
Type:
Small organic molecule
Emp. Form.:
C181H278N54O55
Mol. Mass.:
4090.4728
SMILES:
n/a
Structure:
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