Reaction Details Report a problem with these data
Target
5-hydroxytryptamine receptor 1B
Ligand
BDBM85097
Substrate
n/a
Ki
398.1±n/a nM
Comments
PDSP_1670
Citation
Kennett, GA; Wood, MD; Bright, F; Trail, B; Riley, G; Holland, V; Avenell, KY; Stean, T; Upton, N; Bromidge, S; Forbes, IT; Brown, AM; Middlemiss, DN; Blackburn, TP SB 242084, a selective and brain penetrant 5-HT2C receptor antagonist. Neuropharmacology 36:609-20 (1997) [PubMed] Article
More Info.:
Target
Name:
5-hydroxytryptamine receptor 1B
Synonyms:
5-HT1B | 5-hydroxytryptamine receptor 1A (5HT1B) | 5-hydroxytryptamine receptor 1B (5HT1B) | 5HT1B_CRIGR | HTR1B
Type:
Protein
Mol. Mass.:
42909.60
Organism:
Cricetulus griseus (Chinese hamster) (Cricetulus barabensis griseus)
Description:
P46636
Residue:
386
Sequence:
MEEQGIQCAPPPPAASQTGVPLVNLSHNCSAESHIYQDSIALPWKVLLVALLALITLATTLSNAFVIATVYRTRKLHTPANYLIASLAVTDLLVSILVMPVSTMYTVTGRWTLGQVVCDFWLSSDITCCTASIMHLCVIALDRYWAITDAVEYAAKRTPKRAAIMIALVWVFSISISLPPFFWRQAKAEEEVLTCLVNTDHVLYTVYSTGGAFYLPTLLLIALYGRIYVEARSRILKQTPNKTGKRLTRAQLITDSPGSTTSVTSINSRAPDLPSESGSPVYVNQVKVRVSDALLEKKKLMAARERKATKTLGIILGAFIVCWLPFFIISLVMPICKDACWFHMATLDFFNWLGYLNSLINPIIYTMSNEDFKQAFHKLIRFKCAG