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Target
Delta-type opioid receptor
Ligand
BDBM85329
Substrate
n/a
Ki
60.5±n/a nM
Comments
PDSP_1362
Citation
 Toll, L; Berzetei-Gurske, IP; Polgar, WE; Brandt, SR; Adapa, ID; Rodriguez, L; Schwartz, RW; Haggart, D; O'Brien, A; White, A; Kennedy, JM; Craymer, K; Farrington, L; Auh, JS Standard binding and functional assays related to medications development division testing for potential cocaine and opiate narcotic treatment medications. NIDA Res Monogr 178:440-66 (1998) [PubMed] 
Target
Name:
Delta-type opioid receptor
Synonyms:
Delta opioid receptor | Delta-type opioid receptor | OPIATE Delta | OPRD1 | OPRD_PIG
Type:
Enzyme Catalytic Domain
Mol. Mass.:
25736.90
Organism:
GUINEA PIG
Description:
OPIATE Delta OPRD1 GUINEA PIG::P79291
Residue:
228
Sequence:
GIVRYTKMKTATNIYIFNLALADALATSTLPFQSAKYLMETWPFGELLCKAVLSIDYYNMFTSIFTLTMMSVDRYIAVCHPVKALDFRTPAKAKLINICIWVLASGVGVPIMVMAVTRPRDGAVVCMLQFPSPSWYWDTVTKICVFLFAFVVPILVITVCYGLMLLRLRSVRLLSGSKEKDRSLRRITRMVLVVVGAFVVCWAPIHIFVIVWTLVDIDRRDPLVVAAL
  
Inhibitor
Name:
BDBM85329
Synonyms:
NORMORPHINE
Type:
Small organic molecule
Emp. Form.:
C16H17NO3
Mol. Mass.:
271.3111
SMILES:
[H]C12Cc3ccc(O)c4OC5C(O)C=CC1C5(CCN2)c34 |c:13,TLB:8:20:15:19.17.18|
Structure:
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