Target
Neuropeptide Y receptor type 2
Ligand
BDBM82276
Substrate
n/a
Ki
366±n/a nM
Comments
PDSP_7555
Citation
 Sharma, PHolmberg, SKEriksson, HBeck-Sickinger, AGGrundemar, LLarhammar, D Cloning and functional expression of the guinea pig neuropeptide Y Y2 receptor. Regul Pept 0:23-8 (1998) [PubMed]  Article 
Target
Name:
Neuropeptide Y receptor type 2
Synonyms:
NPY-Y2 | NPY2R | NPY2R_CAVPO | Neuropeptide Y receptor type 2
Type:
Enzyme Catalytic Domain
Mol. Mass.:
42344.53
Organism:
GUINEA PIG
Description:
NPY-Y2 NPY2R GUINEA PIG::Q9Z2D5
Residue:
381
Sequence:
MGPIGTEADENQTVEEIKVEPYGPGHTTPRGELAPDPEPELIDSTKLTEVRVVLILAYCSIILLGVVGNSLVIHVVIKFKSMRTVTNFFIANLAVADLLVNTLCLPFTLTYTLMGEWKMGPVLCHLVPYAQGLAVQVSTVTLTVIALDRHRCIVYHLDSKISKQNSFLIIGLAWGISALLASPLAIFREYSLIEIIPDFEIVACTEKWPGEEKSIYGTVYSLSSLLILYVLPLGIISVSYVRIWSKLKNHVSPGAANDHYHQRRQKTTKMLVFVVVVFAVSWLPLHAFQLAVDIDSQVLDLKEYKLIFTVFHIIAMCSTFANPLLYGWMNSNYRKAFLSAFRCQQRLDAIQSEVCVTGKAKTNVEVEKNHGAADSAEATNV
  
Inhibitor
Name:
BDBM82276
Synonyms:
L31,P34-NPY,human | NPY Leu31, Pro34, human, rat | NPY [Leu31, Pro34], human | NPY, LP, porcine | NPY,[Leu31,Pro34] | NPY,[leu31,Pro34], porcine
Type:
Small organic molecule
Emp. Form.:
C188H282N54O56S
Mol. Mass.:
4226.644
SMILES:
n/a
Structure:
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