Target
Galanin receptor type 2
Ligand
BDBM85072
Substrate
n/a
Ki
2.34±n/a nM
Comments
PDSP_864
Citation
 Borowsky, BWalker, MWHuang, LYJones, KASmith, KEBard, JBranchek, TAGerald, C Cloning and characterization of the human galanin GALR2 receptor. Peptides 19:1771-81 (1998) [PubMed]  Article 
Target
Name:
Galanin receptor type 2
Synonyms:
Galanin receptor type 2 (GAL2-R) (GALR2). | Galanin receptor 2 | Galanin R2 | Galanin receptor type 2 | GALR2_HUMAN | GALR2 | GALNR2
Type:
Enzyme Catalytic Domain
Mol. Mass.:
41724.40
Organism:
Human
Description:
Galanin R2 GALR2 HUMAN::O43603
Residue:
387
Sequence:
MNVSGCPGAGNASQAGGGGGWHPEAVIVPLLFALIFLVGTVGNTLVLAVLLRGGQAVSTTNLFILNLGVADLCFILCCVPFQATIYTLDGWVFGSLLCKAVHFLIFLTMHASSFTLAAVSLDRYLAIRYPLHSRELRTPRNALAAIGLIWGLSLLFSGPYLSYYRQSQLANLTVCHPAWSAPRRRAMDICTFVFSYLLPVLVLGLTYARTLRYLWRAVDPVAAGSGARRAKRKVTRMILIVAALFCLCWMPHHALILCVWFGQFPLTRATYALRILSHLVSYANSCVNPIVYALVSKHFRKGFRTICAGLLGRAPGRASGRVCAAARGTHSGSVLERESSDLLHMSEAAGALRPCPGASQPCILEPCPGPSWQGPKAGDSILTVDVA
  
Inhibitor
Name:
BDBM85072
Synonyms:
Galanin, Human
Type:
Small organic molecule
Emp. Form.:
TBD
Mol. Mass.:
TBD
SMILES:
TBD
Structure:
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