Reaction Details Report a problem with these data
Target
Somatostatin receptor type 1
Ligand
BDBM50232821
Substrate
n/a
Ki
3.3±n/a nM
Comments
PDSP_3372
Citation
 Patel, YC Somatostatin and its receptor family. Front Neuroendocrinol 20:157-98 (1999) [PubMed]  Article 
Target
Name:
Somatostatin receptor type 1
Synonyms:
SOMATOSTATIN SST1 | SRIF-2 | SS-1-R | SS1-R | SS1R | SSR1_HUMAN | SSTR1 | Somatostatin receptor type 1 (SSTR1)
Type:
Enzyme
Mol. Mass.:
42692.81
Organism:
Homo sapiens (Human)
Description:
P30872
Residue:
391
Sequence:
MFPNGTASSPSSSPSPSPGSCGEGGGSRGPGAGAADGMEEPGRNASQNGTLSEGQGSAILISFIYSVVCLVGLCGNSMVIYVILRYAKMKTATNIYILNLAIADELLMLSVPFLVTSTLLRHWPFGALLCRLVLSVDAVNMFTSIYCLTVLSVDRYVAVVHPIKAARYRRPTVAKVVNLGVWVLSLLVILPIVVFSRTAANSDGTVACNMLMPEPAQRWLVGFVLYTFLMGFLLPVGAICLCYVLIIAKMRMVALKAGWQQRKRSERKITLMVMMVVMVFVICWMPFYVVQLVNVFAEQDDATVSQLSVILGYANSCANPILYGFLSDNFKRSFQRILCLSWMDNAAEEPVDYYATALKSRAYSVEDFQPENLESGGVFRNGTCTSRITTL
  
Inhibitor
Name:
BDBM50232821
Synonyms:
(S)-((S)-2-aminopropyl) 6-amino-2-(2-(2-(naphthalen-2-yl)-1H-benzo[g]indol-3-yl)acetamido)hexanoate | CHEMBL252764 | L-817,818
Type:
Small organic molecule
Emp. Form.:
C33H36N4O3
Mol. Mass.:
536.6639
SMILES:
C[C@H](N)COC(=O)[C@H](CCCCN)NC(=O)Cc1c([nH]c2c1ccc1ccccc21)-c1ccc2ccccc2c1
Structure:
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