Ki Summary

Reaction Details

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Target

Somatostatin receptor type 3

Ligand

BDBM81767

Substrate

n/a

0.3±n/a nM

Comments

PDSP_1735

Citation

Patel, YC Somatostatin and its receptor family. Front Neuroendocrinol 20:157-98 (1999) [PubMed] Article

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Target

Name:

Somatostatin receptor type 3

Synonyms:

SSR-28 | SS-3-R | SS3-R | Somatostatin receptor type 3 (SSTR3) | SOMATOSTATIN SST3 | SS3R | SSR3_HUMAN | SSTR3

Type:

Protein

Mol. Mass.:

45855.97

Organism:

Human

Description:

P32745

Residue:

418

Sequence:

MDMLHPSSVSTTSEPENASSAWPPDATLGNVSAGPSPAGLAVSGVLIPLVYLVVCVVGLLGNSLVIYVVLRHTASPSVTNVYILNLALADELFMLGLPFLAAQNALSYWPFGSLMCRLVMAVDGINQFTSIFCLTVMSVDRYLAVVHPTRSARWRTAPVARTVSAAVWVASAVVVLPVVVFSGVPRGMSTCHMQWPEPAAAWRAGFIIYTAALGFFGPLLVICLCYLLIVVKVRSAGRRVWAPSCQRRRRSERRVTRMVVAVVALFVLCWMPFYVLNIVNVVCPLPEEPAFFGLYFLVVALPYANSCANPILYGFLSYRFKQGFRRVLLRPSRRVRSQEPTVGPPEKTEEEDEEEEDGEESREGGKGKEMNGRVSQITQPGTSGQERPPSRVASKEQQLLPQEASTGEKSSTMRISYL

Inhibitor

Name:

BDBM81767

Synonyms:

15-28-Somatostatin-28 | CB6417646 | CAS_38916-34-6 | Somatostatin-14

Type:

Small organic molecule

Emp. Form.:

n/a

Mol. Mass.:

n/a

SMILES:

C[C@@H](O)[C@@H]1NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CSSC[C@H](NC(=O)[C@H](CO)NC1=O)C(O)=O)NC(=O)CNC(=O)[C@H](C)N)[C@@H](C)O |r|

Structure: