Reaction Details Report a problem with these data
Target
Somatostatin receptor type 4
Ligand
BDBM50063821
Substrate
n/a
Ki
66±n/a nM
Comments
PDSP_3363
Citation
 Patel, YC Somatostatin and its receptor family. Front Neuroendocrinol 20:157-98 (1999) [PubMed]  Article 
Target
Name:
Somatostatin receptor type 4
Synonyms:
SOMATOSTATIN SST4 | SS-4-R | SS4-R | SS4R | SSR4_HUMAN | SST4R | SSTR4 | Somatostatin receptor type 4 (SSTR4)
Type:
Enzyme
Mol. Mass.:
42015.38
Organism:
Homo sapiens (Human)
Description:
P31391
Residue:
388
Sequence:
MSAPSTLPPGGEEGLGTAWPSAANASSAPAEAEEAVAGPGDARAAGMVAIQCIYALVCLVGLVGNALVIFVILRYAKMKTATNIYLLNLAVADELFMLSVPFVASSAALRHWPFGSVLCRAVLSVDGLNMFTSVFCLTVLSVDRYVAVVHPLRAATYRRPSVAKLINLGVWLASLLVTLPIAIFADTRPARGGQAVACNLQWPHPAWSAVFVVYTFLLGFLLPVLAIGLCYLLIVGKMRAVALRAGWQQRRRSEKKITRLVLMVVVVFVLCWMPFYVVQLLNLFVTSLDATVNHVSLILSYANSCANPILYGFLSDNFRRFFQRVLCLRCCLLEGAGGAEEEPLDYYATALKSKGGAGCMCPPLPCQQEALQPEPGRKRIPLTRTTTF
  
Inhibitor
Name:
BDBM50063821
Synonyms:
CHEMBL414254 | H-DNal-cyclo[Cys-Tyr-DTrp-Lys-Val-DCys]-Thr-NH2 | H-DNal-cyclo[DCys-Tyr-DTrp-Lys-Val-Cys]-Thr-NH2 | Lanreotide
Type:
Small organic molecule
Emp. Form.:
C54H69N11O10S2
Mol. Mass.:
1096.323
SMILES:
CC(C)[C@@H]1NC(=O)[C@@H](CCCCN)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@@H](Cc2ccc(O)cc2)NC(=O)[C@@H](CSSC[C@H](NC1=O)C(=O)N[C@@H](C(C)O)C(N)=O)NC(=O)[C@H](N)Cc1ccc2ccccc2c1
Structure:
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