Target
Neuropeptide Y receptor type 2
Ligand
BDBM84997
Substrate
n/a
Ki
29±n/a nM
Comments
PDSP_1373
Citation
 Cabrele, CLanger, MBader, RWieland, HADoods, HNZerbe, OBeck-Sickinger, AG The first selective agonist for the neuropeptide YY5 receptor increases food intake in rats. J Biol Chem 275:36043-8 (2000) [PubMed]  Article 
Target
Name:
Neuropeptide Y receptor type 2
Synonyms:
NPY-Y2 | NPY-Y2 receptor | NPY2-R | NPY2R | NPY2R_HUMAN | Neuropeptide Y receptor type 2 | Y2 receptor | neuropeptide Y receptor Y2
Type:
Enzyme Catalytic Domain
Mol. Mass.:
42734.65
Organism:
Homo sapiens (Human)
Description:
NPY-Y2 NPY2R HUMAN::P49146
Residue:
381
Sequence:
MGPIGAEADENQTVEEMKVEQYGPQTTPRGELVPDPEPELIDSTKLIEVQVVLILAYCSIILLGVIGNSLVIHVVIKFKSMRTVTNFFIANLAVADLLVNTLCLPFTLTYTLMGEWKMGPVLCHLVPYAQGLAVQVSTITLTVIALDRHRCIVYHLESKISKRISFLIIGLAWGISALLASPLAIFREYSLIEIIPDFEIVACTEKWPGEEKSIYGTVYSLSSLLILYVLPLGIISFSYTRIWSKLKNHVSPGAANDHYHQRRQKTTKMLVCVVVVFAVSWLPLHAFQLAVDIDSQVLDLKEYKLIFTVFHIIAMCSTFANPLLYGWMNSNYRKAFLSAFRCEQRLDAIHSEVSVTFKAKKNLEVRKNSGPNDSFTEATNV
  
Inhibitor
Name:
BDBM84997
Synonyms:
NPY D-Trp32 | NPY D-Trp32, human, rat | NPY D-Trp32, porcine
Type:
Small organic molecule
Emp. Form.:
C196H290N56O56S
Mol. Mass.:
4358.806
SMILES:
n/a
Structure:
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