Reaction Details Report a problem with these data
Target
Cannabinoid receptor 1
Ligand
BDBM85675
Substrate
n/a
Ki
2795±n/a nM
Comments
PDSP_3416
Citation
 Soderstrom, K; Johnson, F Zebra finch CB1 cannabinoid receptor: pharmacology and in vivo and in vitro effects of activation. J Pharmacol Exp Ther 297:189-97 (2001) [PubMed] 
Target
Name:
Cannabinoid receptor 1
Synonyms:
CANNABINOID CB1 | CNR1 | CNR1_TAEGU
Type:
Enzyme Catalytic Domain
Mol. Mass.:
53103.29
Organism:
Zebra Finch
Description:
CANNABINOID CB1 CNR1 Zebra Finch::P56971
Residue:
473
Sequence:
MKSILDGLADTTFRTITTDLLYVGSNDIQYEDMKGDMASKLGYYPQKFPLSSFRGDPFQEKMTGGDDSLLSIIPSEQVNITEFYNKSLSTFKDNEENIQCGENFMDMECFMILNPSQQLAIAVLSLTLGTFTVLENLLVLCVILHSRSLRCRPSYHFIGSLAVADLLGSVIFVYSFVDFHVFHRKDSPNVFLFKLGGVTASFTASVGSLFLTAIDRYISIHRPLAYKRIVTRPKAVVAFCVMWTIAIVIAVLPLLGWNCKKLNSVCSDIFPLIDETYLMFWIGVTSILLLFIVYAYMYILWKAHSHAVRMLQRGTQKSIIIQSTEDGKVQITRPDQTRMDIRLAKTLVLILVVLIICWGPLLAIMVYDVFGKMNKLIKTIFAFCSMLCLLNSTVNPIIYALRSKDLRHAFRSMFPTCEGTAQPLDNSMESDCQHKHANNAGNVHRAAESCIKSTVKIAKVTMSVSTDTTAEAL
  
Inhibitor
Name:
BDBM85675
Synonyms:
Anandamide + PMSF | CHEMBL321585
Type:
Small organic molecule
Emp. Form.:
C24H41NO2
Mol. Mass.:
375.5878
SMILES:
CCCCC\C=C/C\C=C/C\C=C/C\C=C/CCCCCC(=O)NCCO
Structure:
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