Target
Neuropeptide Y receptor type 1
Ligand
BDBM82287
Substrate
n/a
Ki
24.55±n/a nM
Comments
PDSP_1389
Citation
 Holmberg, SKMikko, SBoswell, TZoorob, RLarhammar, D Pharmacological characterization of cloned chicken neuropeptide Y receptors Y1 and Y5. J Neurochem 81:462-71 (2002) [PubMed]  Article 
Target
Name:
Neuropeptide Y receptor type 1
Synonyms:
NPY-Y1 | NPY1R | Neuropeptide Y receptor Y1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
44370.70
Organism:
Chicken
Description:
Q8QFM1
Residue:
385
Sequence:
MNASVLDPLGNNSSHLNFSEKNSQILQFEDEDCHVPLAMVFTLALAYGTVIILGVSGNLALIVIILKQKEMRNVTNILIVNLSFSDLLVTIMCLPFTFVYTLMDHWIFGEAMCKLNPFVQCASITVSVFSLVLIAIERHQLIINPRGWRPNNRHAYMGIAAIWVLATASSLPFLIYHVLTDEPFRNITFDEYKDKYVCLDLFPLDTARLSYTTTLLVIQYFGPLCFIFICYLKIYFRLKKRSNMMDKMRDSKYRSSETKRINIMLISIVVAFAVCWLPLTIFNIVFDWNHEILPVATCSHNLLFLICHLTAMISTCVNPIFYGFLNKNFQRDLQFLFHFCHFRSREEDYETIAMSTMHTDVSKTSLKQASPVAFKKINSDDDDKI
  
Inhibitor
Name:
BDBM82287
Synonyms:
NPY2-36 | NPY2-36, human | NPY2-36, porcine
Type:
Small organic molecule
Emp. Form.:
C181H278N54O55
Mol. Mass.:
4090.4728
SMILES:
n/a
Structure:
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