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Target
Mu-type opioid receptor
Ligand
BDBM86056
Substrate
n/a
Ki
0.25±n/a nM
Comments
PDSP_2985
Citation
 Gharagozlou, P; Demirci, H; David Clark, J; Lameh, J Activity of opioid ligands in cells expressing cloned mu opioid receptors. BMC Pharmacol 3:1 (2003) [PubMed]  Article 
Target
Name:
Mu-type opioid receptor
Synonyms:
M-OR-1 | MOP | MOR-1 | MOR1 | MUOR1 | Mu Opioid Receptor | Mu opiate receptor | OPIATE Mu | OPRM1 | OPRM_HUMAN | hMOP | mu-type opioid receptor isoform MOR-1
Type:
G Protein-Coupled Receptor (GPCR)
Mol. Mass.:
44789.51
Organism:
Homo sapiens (Human)
Description:
P35372
Residue:
400
Sequence:
MDSSAAPTNASNCTDALAYSSCSPAPSPGSWVNLSHLDGNLSDPCGPNRTDLGGRDSLCPPTGSPSMITAITIMALYSIVCVVGLFGNFLVMYVIVRYTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSIFTLCTMSVDRYIAVCHPVKALDFRTPRNAKIINVCNWILSSAIGLPVMFMATTKYRQGSIDCTLTFSHPTWYWENLLKICVFIFAFIMPVLIITVCYGLMILRLKSVRMLSGSKEKDRNLRRITRMVLVVVAVFIVCWTPIHIYVIIKALVTIPETTFQTVSWHFCIALGYTNSCLNPVLYAFLDENFKRCFREFCIPTSSNIEQQNSTRIRQNTRDHPSTANTVDRTNHQLENLEAETAPLP
  
Inhibitor
Name:
BDBM86056
Synonyms:
CAS_156889 | NSC_156889 | Xorphanol
Type:
Small organic molecule
Emp. Form.:
C23H31NO
Mol. Mass.:
337.4983
SMILES:
CC1CC(=C)CC23CCN(CC4CCC4)C(Cc4ccc(O)cc24)C13 |THB:1:24:16.17.23:9.8.7,10:9:24:16.17.23,22:23:24:9.8.7|
Structure:
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