Reaction Details Report a problem with these data
Target
Hrh3 protein
Ligand
BDBM86057
Substrate
n/a
Ki
>10000±n/a nM
Comments
PDSP_3030
Citation
 Hameg, A; Bayle, F; Nuss, P; Dupuis, P; Garay, RP; Dib, M Affinity of cyamemazine, an anxiolytic antipsychotic drug, for human recombinant dopamine vs. serotonin receptor subtypes. Biochem Pharmacol 65:435-40 (2003) [PubMed]  Article 
Target
Name:
Hrh3 protein
Synonyms:
HISTAMINE H3 | HRH3 | Hrh3 protein
Type:
Enzyme Catalytic Domain
Mol. Mass.:
37860.96
Organism:
RAT
Description:
Q5PPG3
Residue:
344
Sequence:
MERAPPDGLMNASGTLAGEAAAAGGARGFSAAWTAVLAALMALLIVATVLGNALVMLAFVADSSLRTQNNFFLLNLAISDFLVGAFCIPLYVPYVLTGRWTFGRGLCKLWLVVDYLLCASSVFNIVLISYDRFLSVTRAVSYRAQQGDTRRAVRKMALVWVLAFLLYGPAILSWEYLSGGSSIPEGHCYAEFFYNWYFLITASTLEFFTPFLSVTFFNLSIYLNIQRRTRLRLDGGREAGPEPPPDAQPSPPPAPPSCWGCWPKGHGEAMPLHRGSKPSASSASLEKRMKMVSQSITQRFRLSRDKKVAKSLAIIVSIFGLCWAPYTLLMIIRAACHGRCIPDY
  
Inhibitor
Name:
BDBM86057
Synonyms:
CAS_62865 | Cyamemazine | NSC_62865
Type:
Small organic molecule
Emp. Form.:
C19H21N3S
Mol. Mass.:
323.455
SMILES:
CC(CN(C)C)CN1c2ccccc2Sc2ccc(cc12)C#N
Structure:
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