Reaction Details Report a problem with these data
Target
Matrix metalloproteinase-14 [1-20,P8S]
Ligand
BDBM92489
Substrate
n/a
Meas. Tech.
Inhibition Assay
Temperature
310.15±0 K
IC50
>1.00e+5±n/a nM
Citation
 Radichev, IA; Remacle, AG; Shiryaev, SA; Purves, AN; Johnson, SL; Pellecchia, M; Strongin, AY Biochemical characterization of the cellular glycosylphosphatidylinositol-linked membrane type-6 matrix metalloproteinase. J Biol Chem 285:16076-86 (2010) [PubMed]  Article 
Target
Name:
Matrix metalloproteinase-14 [1-20,P8S]
Synonyms:
MMP-14 | MMP-X1 | MMP14 | MMP14_HUMAN | MT-MMP 1 | MT1-MMP | MT1MMP | MTMMP1 | Matrix metalloproteinase 14 | Matrix metalloproteinase-14 | Membrane-type matrix metalloproteinase 1 | Membrane-type-1 matrix metalloproteinase
Type:
Protein
Mol. Mass.:
2138.64
Organism:
Homo sapiens (Human)
Description:
Q8IXG1
Residue:
20
Sequence:
MSPAPRPSRCLLLPLLTLGT
  
Inhibitor
Name:
BDBM92489
Synonyms:
BI-102C8
Type:
Small organic molecule
Emp. Form.:
C15H15NO3
Mol. Mass.:
257.2845
SMILES:
CCOc1ccc(cc1)-c1ccccc1C(=O)NO
Structure:
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