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Target
Calcium/calmodulin-dependent protein kinase II inhibitor 2
Ligand
BDBM50011236
Substrate
n/a
Meas. Tech.
Enzyme Assay
pH
7.4±0
Temperature
303.15±0 K
IC50
5.8e+4±n/a nM
Citation
 Chijiwa, T; Hagiwara, M; Hidaka, H A newly synthesized selective casein kinase I inhibitor, N-(2-aminoethyl)-5-chloroisoquinoline-8-sulfonamide, and affinity purification of casein kinase I from bovine testis. J Biol Chem 264:4924-7 (1989) [PubMed] 
Target
Name:
Calcium/calmodulin-dependent protein kinase II inhibitor 2
Synonyms:
CAMK2N2 | CK2N2_BOVIN | CaM-KII | Calcium/calmodulin-dependent protein kinase II
Type:
Protein
Mol. Mass.:
8656.67
Organism:
Bos taurus (Bovine)
Description:
A5D7T0
Residue:
79
Sequence:
MSEILPYSEDKMGRFGADPEGSDLSFSCRLQDTNSFFAGNQAKRPPKLGQIGRAKRVVIEDDRIDDVLKGMGEKPPSGV
  
Inhibitor
Name:
BDBM50011236
Synonyms:
CHEMBL344314 | Isoquinoline-5-sulfonic acid (2-amino-ethyl)-amide | Isoquinolinesulfonamide, H-9 | N-(2-aminoethyl)isoquinoline-5-sulfonamide
Type:
Small organic molecule
Emp. Form.:
C11H13N3O2S
Mol. Mass.:
251.305
SMILES:
NCCNS(=O)(=O)c1cccc2cnccc12
Structure:
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