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Target
Calcium/calmodulin-dependent protein kinase II inhibitor 2
Ligand
BDBM92674
Substrate
n/a
Meas. Tech.
Enzyme Assay
pH
7.4±0
Temperature
303.15±0 K
IC50
1.95e+5±n/a nM
Citation
 Chijiwa, T; Hagiwara, M; Hidaka, H A newly synthesized selective casein kinase I inhibitor, N-(2-aminoethyl)-5-chloroisoquinoline-8-sulfonamide, and affinity purification of casein kinase I from bovine testis. J Biol Chem 264:4924-7 (1989) [PubMed] 
Target
Name:
Calcium/calmodulin-dependent protein kinase II inhibitor 2
Synonyms:
CAMK2N2 | CK2N2_BOVIN | CaM-KII | Calcium/calmodulin-dependent protein kinase II
Type:
Protein
Mol. Mass.:
8656.67
Organism:
Bos taurus (Bovine)
Description:
A5D7T0
Residue:
79
Sequence:
MSEILPYSEDKMGRFGADPEGSDLSFSCRLQDTNSFFAGNQAKRPPKLGQIGRAKRVVIEDDRIDDVLKGMGEKPPSGV
  
Inhibitor
Name:
BDBM92674
Synonyms:
Isoquinolinesulfonamide, CKI-7
Type:
Small molecule
Emp. Form.:
C11H12ClN3O2S
Mol. Mass.:
285.75
SMILES:
NCCNS(=O)(=O)c1ccc(Cl)c2ccncc12
Structure:
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