Reaction Details Report a problem with these data
Target
Serine/threonine-protein kinase PAK 4
Ligand
BDBM93207
Substrate
n/a
Meas. Tech.
Fluorescence Assay
pH
7.5000±0.0000
Temperature
298.1500±0.0000 K
IC50
>10000±0.2 nM
Citation
 Brigham, JL; Perera, BG; Maly, DJ A Hexylchloride-Based Catch-and-Release System for Chemical Proteomic Applications. ACS Chem Biol 8:691-9 (2013) [PubMed]  Article 
Target
Name:
Serine/threonine-protein kinase PAK 4
Synonyms:
p21-Activated kinase 4 (PAK4) | PAK4_HUMAN | PAK4 | KIAA1142
Type:
Protein
Mol. Mass.:
64098.01
Organism:
Human
Description:
O96013
Residue:
591
Sequence:
MFGKRKKRVEISAPSNFEHRVHTGFDQHEQKFTGLPRQWQSLIEESARRPKPLVDPACITSIQPGAPKTIVRGSKGAKDGALTLLLDEFENMSVTRSNSLRRDSPPPPARARQENGMPEEPATTARGGPGKAGSRGRFAGHSEAGGGSGDRRRAGPEKRPKSSREGSGGPQESSRDKRPLSGPDVGTPQPAGLASGAKLAAGRPFNTYPRADTDHPSRGAQGEPHDVAPNGPSAGGLAIPQSSSSSSRPPTRARGAPSPGVLGPHASEPQLAPPACTPAAPAVPGPPGPRSPQREPQRVSHEQFRAALQLVVDPGDPRSYLDNFIKIGEGSTGIVCIATVRSSGKLVAVKKMDLRKQQRRELLFNEVVIMRDYQHENVVEMYNSYLVGDELWVVMEFLEGGALTDIVTHTRMNEEQIAAVCLAVLQALSVLHAQGVIHRDIKSDSILLTHDGRVKLSDFGFCAQVSKEVPRRKSLVGTPYWMAPELISRLPYGPEVDIWSLGIMVIEMVDGEPPYFNEPPLKAMKMIRDNLPPRLKNLHKVSPSLKGFLDRLLVRDPAQRATAAELLKHPFLAKAGPPASIVPLMRQNRTR
  
Inhibitor
Name:
BDBM93207
Synonyms:
Kinase inhibitor, 5
Type:
Small molecule
Emp. Form.:
TBD
Mol. Mass.:
TBD
SMILES:
TBD
Structure:
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