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Target
Guanine nucleotide-binding protein subunit alpha-15
Ligand
BDBM96755
Substrate
n/a
EC50
24861±n/a nM
Citation
 PubChem, PC Counterscreen for agonists of the human trace amine associated receptor 1 (TAAR1): Fluorescence-based cell-based high throughput dose response assay to identify nonselective Ga16 agonists PubChem Bioassay (2013)[AID] 
Target
Name:
Guanine nucleotide-binding protein subunit alpha-15
Synonyms:
G protein alpha 16 | G-protein subunit alpha-16 | G-protein subunit alpha-16 (G alpha-16) | GNA15 | GNA15_HUMAN | GNA16 | Guanine nucleotide-binding protein subunit alpha-15 [Y147C]
Type:
Protein
Mol. Mass.:
43577.62
Organism:
Homo sapiens (Human)
Description:
P30679
Residue:
374
Sequence:
MARSLTWRCCPWCLTEDEKAAARVDQEINRILLEQKKQDRGELKLLLLGPGESGKSTFIKQMRIIHGAGYSEEERKGFRPLVYQNIFVSMRAMIEAMERLQIPFSRPESKHHASLVMSQDPYKVTTFEKRYAAAMQWLWRDAGIRACYERRREFHLLDSAVYYLSHLERITEEGYVPTAQDVLRSRMPTTGINEYCFSVQKTNLRIVDVGGQKSERKKWIHCFENVIALIYLASLSEYDQCLEENNQENRMKESLALFGTILELPWFKSTSVILFLNKTDILEEKIPTSHLATYFPSFQGPKQDAEAAKRFILDMYTRMYTGCVDGPEGSKKGARSRRLFSHYTCATDTQNIRKVFKDVRDSVLARYLDEINLL
  
Inhibitor
Name:
BDBM96755
Synonyms:
7-Methyl-3-[(2-m-tolyl-ethylamino)-methyl]-1H-quinolin-2-one | 7-methyl-3-[[2-(3-methylphenyl)ethylamino]methyl]-1H-quinolin-2-one | 7-methyl-3-[[2-(m-tolyl)ethylamino]methyl]carbostyril | MLS001209118 | SMR000503418 | cid_3176403
Type:
Small organic molecule
Emp. Form.:
C20H22N2O
Mol. Mass.:
306.4015
SMILES:
Cc1cccc(CCNCc2cc3ccc(C)cc3[nH]c2=O)c1
Structure:
Search PDB for entries with ligand similarity: