Reaction Details Report a problem with these data
Target
Trace amine-associated receptor 1
Ligand
BDBM65923
Substrate
n/a
EC50
674.69±n/a nM
Citation
 PubChem, PC Fluorescence-based cell-based high throughput dose response assay to identify agonists of the human trace amine associated receptor 1 (TAAR1) PubChem Bioassay (2013)[AID] 
Target
Name:
Trace amine-associated receptor 1
Synonyms:
TA1 | TAAR1 | TAAR1_HUMAN | TAR1 | TRAR1 | trace amine-associated receptor 1
Type:
PROTEIN
Mol. Mass.:
39107.47
Organism:
Homo sapiens (Human)
Description:
ChEMBL_792734
Residue:
339
Sequence:
MMPFCHNIINISCVKNNWSNDVRASLYSLMVLIILTTLVGNLIVIVSISHFKQLHTPTNWLIHSMATVDFLLGCLVMPYSMVRSAEHCWYFGEVFCKIHTSTDIMLSSASIFHLSFISIDRYYAVCDPLRYKAKMNILVICVMIFISWSVPAVFAFGMIFLELNFKGAEEIYYKHVHCRGGCSVFFSKISGVLTFMTSFYIPGSIMLCVYYRIYLIAKEQARLISDANQKLQIGLEMKNGISQSKERKAVKTLGIVMGVFLICWCPFFICTVMDPFLHYIIPPTLNDVLIWFGYLNSTFNPMVYAFFYPWFRKALKMMLFGKIFQKDSSRCKLFLELSS
  
Inhibitor
Name:
BDBM65923
Synonyms:
1-(3-Fluoro-phenyl)-3-pyridin-3-yl-urea | 1-(3-fluorophenyl)-3-(3-pyridinyl)urea | 1-(3-fluorophenyl)-3-(3-pyridyl)urea | 1-(3-fluorophenyl)-3-pyridin-3-yl-urea | 1-(3-fluorophenyl)-3-pyridin-3-ylurea | MLS001201441 | SMR000517146 | cid_853873
Type:
Small organic molecule
Emp. Form.:
C12H10FN3O
Mol. Mass.:
231.2257
SMILES:
Fc1cccc(NC(=O)Nc2cccnc2)c1
Structure:
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