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Target
Guanine nucleotide-binding protein subunit alpha-15
Ligand
BDBM96709
Substrate
n/a
IC50
>29877±n/a nM
Citation
 PubChem, PC Counterscreen for agonists of the human trace amine associated receptor 1 (TAAR1): Fluorescence-based cell-based high throughput dose response assay to identify nonselective Ga16 antagonists PubChem Bioassay (2013)[AID] 
Target
Name:
Guanine nucleotide-binding protein subunit alpha-15
Synonyms:
G protein alpha 16 | G-protein subunit alpha-16 | G-protein subunit alpha-16 (G alpha-16) | GNA15 | GNA15_HUMAN | GNA16 | Guanine nucleotide-binding protein subunit alpha-15 [Y147C]
Type:
Protein
Mol. Mass.:
43577.62
Organism:
Homo sapiens (Human)
Description:
P30679
Residue:
374
Sequence:
MARSLTWRCCPWCLTEDEKAAARVDQEINRILLEQKKQDRGELKLLLLGPGESGKSTFIKQMRIIHGAGYSEEERKGFRPLVYQNIFVSMRAMIEAMERLQIPFSRPESKHHASLVMSQDPYKVTTFEKRYAAAMQWLWRDAGIRACYERRREFHLLDSAVYYLSHLERITEEGYVPTAQDVLRSRMPTTGINEYCFSVQKTNLRIVDVGGQKSERKKWIHCFENVIALIYLASLSEYDQCLEENNQENRMKESLALFGTILELPWFKSTSVILFLNKTDILEEKIPTSHLATYFPSFQGPKQDAEAAKRFILDMYTRMYTGCVDGPEGSKKGARSRRLFSHYTCATDTQNIRKVFKDVRDSVLARYLDEINLL
  
Inhibitor
Name:
BDBM96709
Synonyms:
(phenylmethyl) N'-(propan-2-ylideneamino)carbamimidothioate | 2-benzyl-3-(isopropylideneamino)isothiourea | MLS001032917 | N'-(propan-2-ylideneamino)carbamimidothioic acid (phenylmethyl) ester | SMR000363448 | benzyl N'-(propan-2-ylideneamino)carbamimidothioate | cid_5385994
Type:
Small organic molecule
Emp. Form.:
C11H15N3S
Mol. Mass.:
221.322
SMILES:
[#6]\[#6](-[#6])=[#7]\[#7]=[#6](-[#7])-[#16]-[#6]-c1ccccc1 |w:4.3|
Structure:
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