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Target
Guanine nucleotide-binding protein subunit alpha-15
Ligand
BDBM96745
Substrate
n/a
IC50
>29856±n/a nM
Citation
 PubChem, PC Counterscreen for agonists of the human trace amine associated receptor 1 (TAAR1): Fluorescence-based cell-based high throughput dose response assay to identify nonselective Ga16 antagonists PubChem Bioassay (2013)[AID] 
Target
Name:
Guanine nucleotide-binding protein subunit alpha-15
Synonyms:
G protein alpha 16 | G-protein subunit alpha-16 | G-protein subunit alpha-16 (G alpha-16) | GNA15 | GNA15_HUMAN | GNA16 | Guanine nucleotide-binding protein subunit alpha-15 [Y147C]
Type:
Protein
Mol. Mass.:
43577.62
Organism:
Homo sapiens (Human)
Description:
P30679
Residue:
374
Sequence:
MARSLTWRCCPWCLTEDEKAAARVDQEINRILLEQKKQDRGELKLLLLGPGESGKSTFIKQMRIIHGAGYSEEERKGFRPLVYQNIFVSMRAMIEAMERLQIPFSRPESKHHASLVMSQDPYKVTTFEKRYAAAMQWLWRDAGIRACYERRREFHLLDSAVYYLSHLERITEEGYVPTAQDVLRSRMPTTGINEYCFSVQKTNLRIVDVGGQKSERKKWIHCFENVIALIYLASLSEYDQCLEENNQENRMKESLALFGTILELPWFKSTSVILFLNKTDILEEKIPTSHLATYFPSFQGPKQDAEAAKRFILDMYTRMYTGCVDGPEGSKKGARSRRLFSHYTCATDTQNIRKVFKDVRDSVLARYLDEINLL
  
Inhibitor
Name:
BDBM96745
Synonyms:
1,2-bis[(Z)-(4-fluorobenzylidene)amino]guanidine;hydrochloride | 1,2-bis[(Z)-(4-fluorophenyl)methylideneamino]guanidine;hydrochloride | MLS000974588 | N',2-bis(4-fluorobenzylidene)hydrazinecarboximidohydrazide hydrochloride | SMR000496816 | cid_5344776
Type:
Small organic molecule
Emp. Form.:
C15H13F2N5
Mol. Mass.:
301.294
SMILES:
NC(N=NCc1ccc(F)cc1)=NN=Cc1ccc(F)cc1 |w:3.3,13.13,1.0|
Structure:
Search PDB for entries with ligand similarity: