Reaction Details Report a problem with these data
Target
Steroidogenic factor 1
Ligand
BDBM97213
Substrate
n/a
IC50
>67518±n/a nM
Citation
 PubChem, PC Counterscreen for inhibitors of the orphan nuclear receptor subfamily 0, group B, member 1 (DAX1; NR0B1): Luminescence-based cell-based high throughput dose response assay for nonselective inhibitors/assay artifacts using AP2 mutant SF-1 (NR5A1) Transactivation Assay PubChem Bioassay (2013)[AID] 
Target
Name:
Steroidogenic factor 1
Synonyms:
AD4BP | Adrenal 4-binding protein | FTZF1 | Fushi tarazu factor homolog 1 | NR5A1 | Nuclear receptor subfamily 5 group A member 1 | SF-1 | SF1 | STF-1 | STF1_HUMAN | Steroid hormone receptor Ad4BP
Type:
Nuclear Hormone Receptor
Mol. Mass.:
51643.43
Organism:
Homo sapiens (Human)
Description:
n/a
Residue:
461
Sequence:
MDYSYDEDLDELCPVCGDKVSGYHYGLLTCESCKGFFKRTVQNNKHYTCTESQSCKIDKTQRKRCPFCRFQKCLTVGMRLEAVRADRMRGGRNKFGPMYKRDRALKQQKKAQIRANGFKLETGPPMGVPPPPPPAPDYVLPPSLHGPEPKGLAAGPPAGPLGDFGAPALPMAVPGAHGPLAGYLYPAFPGRAIKSEYPEPYASPPQPGLPYGYPEPFSGGPNVPELILQLLQLEPDEDQVRARILGCLQEPTKSRPDQPAAFGLLCRMADQTFISIVDWARRCMVFKELEVADQMTLLQNCWSELLVFDHIYRQVQHGKEGSILLVTGQEVELTTVATQAGSLLHSLVLRAQELVLQLLALQLDRQEFVCLKFIILFSLDLKFLNNHILVKDAQEKANAALLDYTLCHYPHCGDKFQQLLLCLVEVRALSMQAKEYLYHKHLGNEMPRNNLLIEMLQAKQT
  
Inhibitor
Name:
BDBM97213
Synonyms:
2-ethoxy-6-[2-(2-quinolinyl)vinyl]phenyl acetate | MLS000675659 | SMR000294944 | [2-ethoxy-6-[(E)-2-quinolin-2-ylethenyl]phenyl] acetate | [2-ethoxy-6-[(E)-2-quinolin-2-ylethenyl]phenyl] ethanoate | acetic acid [2-ethoxy-6-[(E)-2-(2-quinolinyl)ethenyl]phenyl] ester | acetic acid [2-ethoxy-6-[(E)-2-(2-quinolyl)vinyl]phenyl] ester | cid_5740248
Type:
Small organic molecule
Emp. Form.:
C21H19NO3
Mol. Mass.:
333.3805
SMILES:
CCOc1cccc(\C=C\c2ccc3ccccc3n2)c1OC(C)=O
Structure:
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