Reaction Details
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Report a problem with these dataTarget
COUP transcription factor 2
Ligand
BDBM97096
Substrate
n/a
IC50
2287±n/a nM
Citation
PubChem, PC Luminescence-based cell-based high throughput dose response assay to identify inhibitors of COUP-TFII (NR2F2) PubChem Bioassay (2013)[AID] More Info.:
Target
Name:
COUP transcription factor 2
Synonyms:
ARP1 | COT2_HUMAN | COUP transcription factor 2 isoform a | NR2F2 | TFCOUP2
Type:
Enzyme Catalytic Domain
Mol. Mass.:
45583.83
Organism:
Homo sapiens (Human)
Description:
gi_14149746
Residue:
414
Sequence:
MAMVVSTWRDPQDEVPGSQGSQASQAPPVPGPPPGAPHTPQTPGQGGPASTPAQTAAGGQGGPGGPGSDKQQQQQHIECVVCGDKSSGKHYGQFTCEGCKSFFKRSVRRNLSYTCRANRNCPIDQHHRNQCQYCRLKKCLKVGMRREAVQRGRMPPTQPTHGQFALTNGDPLNCHSYLSGYISLLLRAEPYPTSRFGSQCMQPNNIMGIENICELAARMLFSAVEWARNIPFFPDLQITDQVALLRLTWSELFVLNAAQCSMPLHVAPLLAAAGLHASPMSADRVVAFMDHIRIFQEQVEKLKALHVDSAEYSCLKAIVLFTSDACGLSDVAHVESLQEKSQCALEEYVRSQYPNQPTRFGKLLLRLPSLRTVSSSVIEQLFFVRLVGKTPIETLIRDMLLSGSSFNWPYMAIQ
Inhibitor
Name:
BDBM97096
Synonyms:
4-chloranyl-3-ethoxy-N-(pyridin-4-ylmethyl)benzenesulfonamide | 4-chloro-3-ethoxy-N-(4-pyridinylmethyl)benzenesulfonamide | 4-chloro-3-ethoxy-N-(4-pyridylmethyl)benzenesulfonamide | 4-chloro-3-ethoxy-N-(pyridin-4-ylmethyl)benzenesulfonamide | MLS000676361 | SMR000301136 | cid_2240759
Type:
Small organic molecule
Emp. Form.:
C14H15ClN2O3S
Mol. Mass.:
326.799
SMILES:
CCOc1cc(ccc1Cl)S(=O)(=O)NCc1ccncc1
Structure:
