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Target
Retinol-binding protein 4
Ligand
BDBM106689
Substrate
n/a
Meas. Tech.
Binding Assay
IC50
790±0.0 nM
Citation
 Kasai, S; Kaku, T; Kamaura, M Heterocyclic compound US Patent  US8586571 Publication Date 11/19/2013 
Target
Name:
Retinol-binding protein 4
Synonyms:
PRBP | Plasma retinol-binding protein | RBP | RBP4 | RET4_HUMAN | Retinol-binding protein 4 | Retinol-binding protein 4 (RBP4) | spa binding assay for rbp4
Type:
Protein
Mol. Mass.:
23008.75
Organism:
Homo sapiens (Human)
Description:
P02753
Residue:
201
Sequence:
MKWVWALLLLAALGSGRAERDCRVSSFRVKENFDKARFSGTWYAMAKKDPEGLFLQDNIVAEFSVDETGQMSATAKGRVRLLNNWDVCADMVGTFTDTEDPAKFKMKYWGVASFLQKGNDDHWIVDTDYDTYAVQYSCRLLNLDGTCADSYSFVFSRDPNGLPPEAQKIVRQRQEELCLARQYRLIVHNGYCDGRSERNLL
  
Inhibitor
Name:
BDBM106689
Synonyms:
US8586571, 121
Type:
Small organic molecule
Emp. Form.:
C23H36N2O5S
Mol. Mass.:
452.607
SMILES:
CCCCCS(=O)(=O)NC(=O)C(=O)N1CCC(COc2ccccc2C(C)(C)C)CC1
Structure:
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