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Target
Retinol-binding protein 4
Ligand
BDBM106692
Substrate
n/a
Meas. Tech.
Binding Assay
IC50
71±0.0 nM
Citation
 Kasai, S; Kaku, T; Kamaura, M Heterocyclic compound US Patent  US8586571 Publication Date 11/19/2013 
Target
Name:
Retinol-binding protein 4
Synonyms:
PRBP | Plasma retinol-binding protein | RBP | RBP4 | RET4_HUMAN | Retinol-binding protein 4 | Retinol-binding protein 4 (RBP4) | spa binding assay for rbp4
Type:
Protein
Mol. Mass.:
23008.75
Organism:
Homo sapiens (Human)
Description:
P02753
Residue:
201
Sequence:
MKWVWALLLLAALGSGRAERDCRVSSFRVKENFDKARFSGTWYAMAKKDPEGLFLQDNIVAEFSVDETGQMSATAKGRVRLLNNWDVCADMVGTFTDTEDPAKFKMKYWGVASFLQKGNDDHWIVDTDYDTYAVQYSCRLLNLDGTCADSYSFVFSRDPNGLPPEAQKIVRQRQEELCLARQYRLIVHNGYCDGRSERNLL
  
Inhibitor
Name:
BDBM106692
Synonyms:
US8586571, 189
Type:
Small organic molecule
Emp. Form.:
C17H22ClNO4
Mol. Mass.:
339.814
SMILES:
CC(C)(C)c1cc(Cl)ccc1OC1CN(C1)C(=O)CCC(O)=O
Structure:
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