Reaction Details Report a problem with these data
Target
Trace amine-associated receptor 1
Ligand
BDBM109384
Substrate
n/a
Meas. Tech.
Radioligand Binding Assay
Ki
0.8±n/a nM
Citation
 Galley, G; Groebke Zbinden, K; Norcross, R; Stalder, H 2-aminooxazolines as TAAR1 ligands US Patent  US8604061 Publication Date 12/10/2013 
Target
Name:
Trace amine-associated receptor 1
Synonyms:
TAAR1_MOUSE | Ta1 | Taar1 | Tar1 | Trace amine receptor 1 (TARR1) | Trace amine-associated receptor 1 (TAAR1) | Trace amine-associated receptor1 | Trar1
Type:
Protein
Mol. Mass.:
37635.41
Organism:
Mus musculus (Mouse)
Description:
Q923Y8
Residue:
332
Sequence:
MHLCHAITNISHRNSDWSREVQASLYSLMSLIILATLVGNLIVIISISHFKQLHTPTNWLLHSMAIVDFLLGCLIMPCSMVRTVERCWYFGEILCKVHTSTDIMLSSASIFHLAFISIDRYCAVCDPLRYKAKINISTILVMILVSWSLPAVYAFGMIFLELNLKGVEELYRSQVSDLGGCSPFFSKVSGVLAFMTSFYIPGSVMLFVYYRIYFIAKGQARSINRTNVQVGLEGKSQAPQSKETKAAKTLGIMVGVFLVCWCPFFLCTVLDPFLGYVIPPSLNDALYWFGYLNSALNPMVYAFFYPWFRRALKMVLLGKIFQKDSSRSKLFL
  
Inhibitor
Name:
BDBM109384
Synonyms:
US8604061, 86
Type:
Small organic molecule
Emp. Form.:
C12H15FN2O2
Mol. Mass.:
238.2581
SMILES:
COc1cc(CC[C@H]2COC(N)=N2)ccc1F |r,c:11|
Structure:
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