Reaction Details
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Target
Cyclin-dependent kinase 2 [F80T]
Ligand
BDBM154577
Substrate
n/a
Meas. Tech.
EMSA
Temperature
576.3±0 K
IC50
7.1e+3±n/a nM
Citation
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More Info.:
Target
Name:
Cyclin-dependent kinase 2 [F80T]
Synonyms:
CDK2 | CDK2_HUMAN | CDKN2 | Cyclin-dependent protein kinase 2 (CDK2 F80T)
Type:
Protein
Mol. Mass.:
33892.10
Organism:
Homo sapiens (Human)
Description:
P24941[F80T]
Residue:
298
Sequence:
MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDTETEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVTEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL