Reaction Details Report a problem with these data
Target
Rhomboid protease GlpG
Ligand
BDBM165194
Substrate
n/a
Meas. Tech.
Activity-based Protein Profiling (ABPP)
pH
7.4±0
Temperature
310.15±0 K
IC50
4.6e+3± 1.0e+3 nM
Citation
Wolf, EV; Zeissler, A; Verhelst, SH Inhibitor Fingerprinting of Rhomboid Proteases by Activity-Based Protein Profiling Reveals Inhibitor Selectivity and Rhomboid Autoprocessing. ACS Chem Biol 10:2325-33 (2015) [PubMed] Article
More Info.:
Target
Name:
Rhomboid protease GlpG
Synonyms:
Rhomboid protease (HiGlpG)
Type:
Protein
Mol. Mass.:
21622.69
Organism:
Haemophilus influenzae (g-Proteobacteria)
Description:
n/a
Residue:
192
Sequence:
MKNFLAQQGKITLILTALCVLIYLAQQLGFEDDIMYLMHYPAYEEQDSEVWRYISHTLVHLSNLHILFNLSWFLIFGGMIERTFGSVKLLMLYVVASAITGYVQNYVSGPAFFGLSGVVYAVLGYVFIRDKLNHHLFDLPEGFFTMLLVGIALGFISPLFGVEMGNAAHISGLIVGLIWGFIDSKLRKNSLE