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Target
Glucose-dependent insulinotropic receptor
Ligand
BDBM180672
Substrate
n/a
Meas. Tech.
AlphaScreen cAMP Assay
pH
7.4±n/a
Temperature
310.15±n/a K
EC50
398±n/a nM
Comments
extracted
Citation
Grauert, M; Bakker, R; Breitfelder, S; Buettner, F; Eickelmann, P; Fox, T; Grundl, M; Lehmann-Lintz, T; Rist, W Benzoxazole- and tetrahydrobenzoxazole-substituted pyridazinones as GPR119 agonists US Patent US8772323 Publication Date 7/8/2014
More Info.:
Target
Name:
Glucose-dependent insulinotropic receptor
Synonyms:
G-protein coupled receptor 119 (GPR119) | GP119_HUMAN | GPR119 | Glucose-dependent insulinotropic receptor
Type:
Protein
Mol. Mass.:
36901.49
Organism:
Human
Description:
Q8TDV5
Residue:
335
Sequence:
MESSFSFGVILAVLASLIIATNTLVAVAVLLLIHKNDGVSLCFTLNLAVADTLIGVAISGLLTDQLSSPSRPTQKTLCSLRMAFVTSSAAASVLTVMLITFDRYLAIKQPFRYLKIMSGFVAGACIAGLWLVSYLIGFLPLGIPMFQQTAYKGQCSFFAVFHPHFVLTLSCVGFFPAMLLFVFFYCDMLKIASMHSQQIRKMEHAGAMAGGYRSPRTPSDFKALRTVSVLIGSFALSWTPFLITGIVQVACQECHLYLVLERYLWLLGVGNSLLNPLIYAYWQKEVRLQLYHMALGVKKVLTSFLLFLSARNCGPERPRESSCHIVTISSSEFDG