Reaction Details Report a problem with these data
Target
3-hydroxyacyl-[acyl-carrier-protein] dehydratase FabZ
Ligand
BDBM24777
Substrate
n/a
Meas. Tech.
FabZ Inhibition Assay
pH
7±n/a
Temperature
298.15±n/a K
IC50
5.4e+3± 1.4e+3 nM
Comments
extracted
Citation
McGillick, BE; Kumaran, D; Vieni, C; Swaminathan, S ß-Hydroxyacyl-acyl Carrier Protein Dehydratase (FabZ) from Francisella tularensis and Yersinia pestis: Structure Determination, Enzymatic Characterization, and Cross-Inhibition Studies. Biochemistry 55:1091-9 (2016) [PubMed] Article
More Info.:
Target
Name:
3-hydroxyacyl-[acyl-carrier-protein] dehydratase FabZ
Synonyms:
beta-Hydroxyacyl-acyl carrier protein dehydratase (FtFabZ)
Type:
Protein
Mol. Mass.:
18151.57
Organism:
Francisella tularensis
Description:
n/a
Residue:
163
Sequence:
MSQFNQNNKQIDVMGIRKILPHRYPFALLDKIVDWSVEDRTIVAQKNVTINEDFFNGHFPDFPVMPGVLIVEAMAQATAILGELMAETLFAHVVEKAGGGRRTFMLAGIDKVRVKRPVVPGDVLVIESRMVKQKNIICTAESVAKVDGQIVCSAELMAAYKDY