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Target
Bromodomain-containing protein 2 [71-194,348-455]
Ligand
BDBM205453
Substrate
n/a
Meas. Tech.
Bromodomains Assay for DiscoveRx Gene Symbol
Ki
0.024±0.0 nM
Citation
Tanaka, M; Roberts, JM; Seo, HS; Souza, A; Paulk, J; Scott, TG; DeAngelo, SL; Dhe-Paganon, S; Bradner, JE Design and characterization of bivalent BET inhibitors. Nat Chem Biol 12:1089-1096 (2016) [PubMed] Article
More Info.:
Target
Name:
Bromodomain-containing protein 2 [71-194,348-455]
Synonyms:
BET bromodomain 2(1,2) (BRD2(1,2)) | BRD2 | BRD2_HUMAN | KIAA9001 | RING3
Type:
n/a
Mol. Mass.:
27418.07
Organism:
Homo sapiens (Human)
Description:
P25440 (BRD2, 71-194 and 348-455)
Residue:
232
Sequence:
KPGRVTNQLQYLHKVVMKALWKHQFAWPFRQPVDAVKLGLPDYHKIIKQPMDMGTIKRRLENNYYWAASECMQDFNTMFTNCYIYNKPTDDIVLMAQTLEKIFLQKVASMPQEEQELVVTIPKNEQLKHCNGILKELLSKKHAAYAWPFYKPVDASALGLHDYHDIIKHPMDLSTVKRKMENRDYRDAQEFAADVRLMFSNCYKYNPPDHDVVAMARKLQDVFEFRYAKMPD