Reaction Details Report a problem with these data
Target
Isoform 2 of Protein mono-ADP-ribosyltransferase PARP3 (Long)
Ligand
BDBM207556
Substrate
n/a
Meas. Tech.
PARP-2 and PARP-3 Enzymatic Assay
IC50
199±n/a nM
Citation
More Info.:
Target
Name:
Isoform 2 of Protein mono-ADP-ribosyltransferase PARP3 (Long)
Synonyms:
ADPRT3 | ADPRTL3 | PARP3 | PARP3_HUMAN | Poly [ADP-ribose] polymerase 3 (PARP-3) | Protein mono-ADP-ribosyltransferase PARP3 (Long)
Type:
Protein
Mol. Mass.:
60847.85
Organism:
Homo sapiens (Human)
Description:
Q9Y6F1-2
Residue:
540
Sequence:
MSLLFLAMAPKPKPWVQTEGPEKKKGRQAGREEDPFRSTAEALKAIPAEKRIIRVDPTCPLSSNPGTQVYEDYNCTLNQTNIENNNNKFYIIQLLQDSNRFFTCWNHWGRVGEVGQSKINHFTRLEDAKKDFEKKFREKTKNNWAERDHFVSHPGKYTLIEVQAEDEAQEAVVKVDRGPVRTVTKRVQPCSLDPATQKLITNIFSKEMFKNTMALMDLDVKKMPLGKLSKQQIARGFEALEALEEALKGPTDGGQSLEELSSHFYTVIPHNFGHSQPPPINSPELLQAKKDMLLVLADIELAQALQAVSEQEKTVEEVPHPLDRDYQLLKCQLQLLDSGAPEYKVIQTYLEQTGSNHRCPTLQHIWKVNQEGEEDRFQAHSKLGNRKLLWHGTNMAVVAAILTSGLRIMPHSGGRVGKGIYFASENSKSAGYVIGMKCGAHHVGYMFLGEVALGREHHINTDNPSLKSPPPGFDSVIARGHTEPDPTQDTELELDGQQVVVPQGQPVPCPEFSSSTFSQSEYLIYQESQCRLRYLLEVHL