Reaction Details Report a problem with these data
Target
TspO-like protein
Ligand
BDBM209867
Substrate
n/a
Meas. Tech.
Tryptophan Fluorescence Assay
Kd
5.05e+3±n/a nM
Citation
 Busch, AW; WareJoncas, Z; Montgomery, BL Tryptophan-Rich Sensory Protein/Translocator Protein (TSPO) from Cyanobacterium Fremyella diplosiphon Binds a Broad Range of Functionally Relevant Tetrapyrroles. Biochemistry 56:73-84 (2017) [PubMed]  Article 
Target
Name:
TspO-like protein
Synonyms:
Tryptophan-rich sensory protein/translocator protein (TSPO)
Type:
Protein
Mol. Mass.:
28330.64
Organism:
Fremyella diplosiphon (Cyanobacterium)
Description:
Q6GZK8
Residue:
251
Sequence:
MTQSNNTGILEKFVNTVMGVKTENQQQPSNTLIATTQALDIRAVLVYKLGTILQIAAMMLALLGMEKLVMLIDKNSHLPSWFSTLLAVLFFALLSIRSRIFSLLDNTRSRKTYDQVIRPRWAPPPLVFPIVWMIIAVLRVISSVLIWQQMHHQFLALPLILFVVHLALGDTWNTIFTVERRLGAAVPVVILGPWLSALVVTAIYWQTNPVAGMIFSFSCIWLTVAAVLVFRIWQLNGSEPLYPLKLTPVEK
  
Inhibitor
Name:
BDBM209867
Synonyms:
3-[18-(2-carboxyethyl)-8,13-diethyl-3,7,12,17-tetramethyl-22,23-dihydroporphyrin-2-yl]propanoic acid | Mesoporphyrin IX
Type:
Small organic molecule
Emp. Form.:
C34H38N4O4
Mol. Mass.:
566.6899
SMILES:
CCc1c(C)c2cc3[nH]c(cc4nc(cc5nc(cc1[nH]2)c(C)c5CCC(O)=O)c(CCC(O)=O)c4C)c(C)c3CC
Structure:
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