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Target
TspO-like protein
Ligand
BDBM209868
Substrate
n/a
Meas. Tech.
Tryptophan Fluorescence Assay
Kd
1.91e+3±n/a nM
Citation
 Busch, AW; WareJoncas, Z; Montgomery, BL Tryptophan-Rich Sensory Protein/Translocator Protein (TSPO) from Cyanobacterium Fremyella diplosiphon Binds a Broad Range of Functionally Relevant Tetrapyrroles. Biochemistry 56:73-84 (2017) [PubMed]  Article 
Target
Name:
TspO-like protein
Synonyms:
Tryptophan-rich sensory protein/translocator protein (TSPO)
Type:
Protein
Mol. Mass.:
28330.64
Organism:
Fremyella diplosiphon (Cyanobacterium)
Description:
Q6GZK8
Residue:
251
Sequence:
MTQSNNTGILEKFVNTVMGVKTENQQQPSNTLIATTQALDIRAVLVYKLGTILQIAAMMLALLGMEKLVMLIDKNSHLPSWFSTLLAVLFFALLSIRSRIFSLLDNTRSRKTYDQVIRPRWAPPPLVFPIVWMIIAVLRVISSVLIWQQMHHQFLALPLILFVVHLALGDTWNTIFTVERRLGAAVPVVILGPWLSALVVTAIYWQTNPVAGMIFSFSCIWLTVAAVLVFRIWQLNGSEPLYPLKLTPVEK
  
Inhibitor
Name:
BDBM209868
Synonyms:
3-[18-(2-carboxyethyl)-8,13-bis(ethenyl)-3,7,12,17-tetramethylporphyrin-21,24-diid-2-yl]propanoic acid;iron(2+) | Haemin | Heme
Type:
Small organic molecule
Emp. Form.:
C34H32N4O4
Mol. Mass.:
560.6434
SMILES:
Cc1c(C=C)c2cc3[n-]c(cc4[n-]c(cc5nc(cc1n2)c(C=C)c5C)c(C)c4CCC(O)=O)c(CCC(O)=O)c3C
Structure:
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