Target
N-acetyltransferase domain-containing protein
Ligand
BDBM213237
Substrate
n/a
Meas. Tech.
Isothermal Titration Calorimetry (ITC)
pH
7.5±0
Temperature
298.15±0 K
Kd
1.653e+5± 9.5e+3 nM
Citation
 Majorek, KAKuhn, MLChruszcz, MAnderson, WFMinor, W Structural, functional, and inhibition studies of a Gcn5-related N-acetyltransferase (GNAT) superfamily protein PA4794: a new C-terminal lysine protein acetyltransferase from pseudomonas aeruginosa. J Biol Chem 288:30223-35 (2013) [PubMed]  Article 
Target
Name:
N-acetyltransferase domain-containing protein
Synonyms:
Gcn5-related N-acetyltransferases (GNAT) superfamily protein PA4794 (PA4794)
Type:
Protein
Mol. Mass.:
17787.24
Organism:
Pseudomonas aeruginosa
Description:
Q9HV14
Residue:
160
Sequence:
MQLSHRPAETGDLETVAGFPQDRDELFYCYPKAIWPFSVAQLAAAIAERRGSTVAVHDGQVLGFANFYQWQHGDFCALGNMMVAPAARGLGVARYLIGVMENLAREQYKARLMKISCFNANAAGLLLYTQLGYQPRAIAERHDPDGRRVALIQMDKPLEP
  
Inhibitor
Name:
BDBM213237
Synonyms:
4-Methylumbelliferyl phosphate
Type:
Small organic molecule
Emp. Form.:
C10H7O6P
Mol. Mass.:
254.1338
SMILES:
Cc1cc(=O)oc2cc(OP([O-])([O-])=O)ccc12
Structure:
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