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Target
Cyclin-dependent kinase 2
Ligand
BDBM8037
Substrate
n/a
Meas. Tech.
OctetRed_Method3
KOFF
1.42E+00 s-1
Citation
 D3R, DD CSAR CDK2-CyclinA D3R 219:0 (2015) [PubMed] 
Target
Name:
Cyclin-dependent kinase 2
Synonyms:
Cyclin-dependent kinase 2 (CDK2) | p33 protein kinase | CDK2-Kinase | Cell division protein kinase 2 | Protein cereblon/Cyclin-dependent kinase 2 | CDK2_HUMAN | CDK2 | CDKN2
Type:
Enzyme Subunit
Mol. Mass.:
33938.17
Organism:
Human
Description:
P24941
Residue:
298
Sequence:
MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDTETEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL
  
Inhibitor
Name:
BDBM8037
Synonyms:
4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-amine | 4-(dimethyl-1,3-thiazol-5-yl)pyrimidin-2-amine, 1 | CS12 | 4-(2,4-Dimethylthiazol-5-yl)pyrimidin-2-ylamine | 2-Anilino-4-(thiazol-5-yl)pyrimidine deriv. 8
Type:
Small organic molecule
Emp. Form.:
TBD
Mol. Mass.:
TBD
SMILES:
TBD
Structure:
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