Reaction Details Report a problem with these data
Target
D(4) dopamine receptor [281-332]
Ligand
BDBM232949
Substrate
n/a
Meas. Tech.
Receptor Binding Assay
pH
7.4±n/a
Temperature
295.15±n/a K
IC50
1.0e+4±n/a nM
Comments
extracted
Citation
 Kogan, V; Lurya, L; Tabachnik, L Heterocyclic compounds and uses thereof in the treatment of sexual disorders US Patent  US9353067 Publication Date 5/31/2016 
Target
Name:
D(4) dopamine receptor [281-332]
Synonyms:
DRD4 | DRD4_HUMAN | Dopamine D4 receptor
Type:
Enzyme
Mol. Mass.:
5036.64
Organism:
Homo sapiens (Human)
Description:
D4.4 (aa 281-332)
Residue:
51
Sequence:
AAPSLPQDPCGPDCAPPAPGLPPDPCGSNCAPPDAVRAAALPPQTPPQTRR
  
Inhibitor
Name:
BDBM232949
Synonyms:
US9353067, L-238
Type:
Small organic molecule
Emp. Form.:
C19H20N4O2
Mol. Mass.:
336.3877
SMILES:
Oc1ccccc1N1CCN(Cc2nc3ccccc3c(=O)[nH]2)CC1
Structure:
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