Reaction Details Report a problem with these data
Target
Cytosol aminopeptidase [33-68,L62W]
Ligand
BDBM234297
Substrate
n/a
Meas. Tech.
Kinetic Inhibition Assay
pH
8.4±0
Temperature
298.15±0 K
Ki
3.64e+3±n/a nM
Citation
 Pícha, J; Liboska, R; Bude?ínský, M; Jirácek, J; Pawelczak, M; Mucha, A Unusual activity pattern of leucine aminopeptidase inhibitors based on phosphorus containing derivatives of methionine and norleucine. J Enzyme Inhib Med Chem 26:155-61 (2011) [PubMed]  Article 
Target
Name:
Cytosol aminopeptidase [33-68,L62W]
Synonyms:
AMPL_PIG | Cytosol aminopeptidase | LAP3 | Leucine aminopeptidase (LAP)
Type:
Enzyme
Mol. Mass.:
4015.44
Organism:
Sus scrofa (Pig)
Description:
P28839[33-68,L62W]
Residue:
36
Sequence:
TKGLVLGIYSKEKEDDAPQFTSAGENFDKWVSGKLR
  
Inhibitor
Name:
BDBM234297
Synonyms:
Met-ψ[P(O)(OH)CH2]-Ala (5)
Type:
Small organic molecule
Emp. Form.:
C8H18NO4PS
Mol. Mass.:
255.272
SMILES:
CSCCC(N)P(O)(=O)CC(C)C(O)=O
Structure:
Search PDB for entries with ligand similarity: