Reaction Details Report a problem with these data
Target
Stimulator of interferon genes protein [H232R]
Ligand
BDBM457783
Substrate
n/a
Meas. Tech.
3H-cGAMP Filtration Binding Assay
EC50
2.40±n/a nM
Citation
Altman, MD; Andresen, B; Chang, W; Childers, ML; Cumming, JN; Haidle, AM; Henderson, TJ; Jewell, JP; Lu, M; Northrup, AB; Otte, RD; Siu, T; Trotter, BW; Truong, QT Cyclic di-nucleotide compounds as STING agonists US Patent US10738074 Publication Date 8/11/2020
More Info.:
Target
Name:
Stimulator of interferon genes protein [H232R]
Synonyms:
ERIS | MITA | STING | STING1 | STING_HUMAN | Stimulator of interferon genes protein STING (H232R) | TMEM173
Type:
Enzyme Catalytic Domain
Mol. Mass.:
42215.19
Organism:
Homo sapiens (Human)
Description:
n/a
Residue:
379
Sequence:
MPHSSLHPSIPCPRGHGAQKAALVLLSACLVTLWGLGEPPEHTLRYLVLHLASLQLGLLLNGVCSLAEELRHIHSRYRGSYWRTVRACLGCPLRRGALLLLSIYFYYSLPNAVGPPFTWMLALLGLSQALNILLGLKGLAPAEISAVCEKGNFNVAHGLAWSYYIGYLRLILPELQARIRTYNQHYNNLLRGAVSQRLYILLPLDCGVPDNLSMADPNIRFLDKLPQQTGDRAGIKDRVYSNSIYELLENGQRAGTCVLEYATPLQTLFAMSQYSQAGFSREDRLEQAKLFCRTLEDILADAPESQNNCRLIAYQEPADDSSFSLSQEVLRHLRQEEKEEVTVGSLKTSAVPSTSTMSQEPELLISGMEKPLPLRTDFS