Reaction Details Report a problem with these data
Target
Isocitrate dehydrogenase [NADP], mitochondrial [40-452,R172K]
Ligand
BDBM50503254
Substrate
n/a
Meas. Tech.
Inhibitory Activity Assay
IC50
22.4±n/a nM
Citation
More Info.:
Target
Name:
Isocitrate dehydrogenase [NADP], mitochondrial [40-452,R172K]
Synonyms:
IDH2 | IDHP_HUMAN | Isocitrate dehydrogenase [NADP], mitochondrial (IDH2) (R172K)
Type:
Enzyme Catalytic Domain
Mol. Mass.:
46594.87
Organism:
Homo sapiens (Human)
Description:
aa 40-end
Residue:
413
Sequence:
ADKRIKVAKPVVEMDGDEMTRIIWQFIKEKLILPHVDIQLKYFDLGLPNRDQTDDQVTIDSALATQKYSVAVKCATITPDEARVEEFKLKKMWKSPNGTIRNILGGTVFREPIICKNIPRLVPGWTKPITIGKHAHGDQYKATDFVADRAGTFKMVFTPKDGSGVKEWEVYNFPAGGVGMGMYNTDESISGFAHSCFQYAIQKKWPLYMSTKNTILKAYDGRFKDIFQEIFDKHYKTDFDKNKIWYEHRLIDDMVAQVLKSSGGFVWACKNYDGDVQSDILAQGFGSLGLMTSVLVCPDGKTIEAEAAHGTVTRHYREHQKGRPTSTNPIASIFAWTRGLEHRGKLDGNQDLIRFAQMLEKVCVETVESGAMTKDLAGCIHGLSNVKLNEHFLNTTDFLDTIKSNLDRALGRQ