Reaction Details Report a problem with these data
Target
Genome polyprotein [1973-2419]
Ligand
BDBM466321
Substrate
n/a
Meas. Tech.
Inhibition Assay
IC50
<1000±n/a nM
Citation
Beigelman, L; Wang, G; Smith, DB Substituted nucleosides, nucleotides and analogs thereof US Patent US10793591 Publication Date 10/6/2020
More Info.:
Target
Name:
Genome polyprotein [1973-2419]
Synonyms:
Non-structural protein 5A (NS5A) | POLG_HCVCO | RNA-directed RNA polymerase (NS5B)
Type:
Enzyme Catalytic Domain
Mol. Mass.:
48705.67
Organism:
Hepatitis C virus genotype 1b (isolate Con1) (HCV)
Description:
Q9WMX2[1973-2419]
Residue:
447
Sequence:
SGSWLRDVWDWICTVLTDFKTWLQSKLLPRLPGVPFFSCQRGYKGVWRGDGIMQTTCPCGAQITGHVKNGSMRIVGPRTCSNTWHGTFPINAYTTGPCTPSPAPNYSRALWRVAAEEYVEVTRVGDFHYVTGMTTDNVKCPCQVPAPEFFTEVDGVRLHRYAPACKPLLREEVTFLVGLNQYLVGSQLPCEPEPDVAVLTSMLTDPSHITAETAKRRLARGSPPSLASSSASQLSAPSLKATCTTRHDSPDADLIEANLLWRQEMGGNITRVESENKVVILDSFEPLQAEEDEREVSVPAEILRRSRKFPRAMPIWARPDYNPPLLESWKDPDYVPPVVHGCPLPPAKAPPIPPPRRKRTVVLSESTVSSALAELATKTFGSSESSAVDSGTATASPDQPSDDGDAGSDVESYSSMPPLEGEPGDPDLSDGSWSTVSEEASEDVVCC