Reaction Details Report a problem with these data
Target
Stimulator of interferon genes protein [139-379,H232R]
Ligand
BDBM501364
Substrate
n/a
Meas. Tech.
STING SPA Binding Assay
IC50
<10.00±n/a nM
Citation
Emanuel, S; Richter, M; Connolly, PJ; Edwards, JP; Wang, G; Thatikonda, SK; Beigelman, L; Zhong, M; Bignan, G Cyclic dinucleotides as sting agonists US Patent US11021511 Publication Date 6/1/2021
More Info.:
Target
Name:
Stimulator of interferon genes protein [139-379,H232R]
Synonyms:
ERIS | MITA | STING | STING1 | STING_HUMAN | Stimulator of interferon genes protein (aa 139-379 H232R) | TMEM173
Type:
Enzyme Catalytic Domain
Mol. Mass.:
27090.78
Organism:
Homo sapiens (Human)
Description:
n/a
Residue:
241
Sequence:
LAPAEISAVCEKGNFNVAHGLAWSYYIGYLRLILPELQARIRTYNQHYNNLLRGAVSQRLYILLPLDCGVPDNLSMADPNIRFLDKLPQQTGDRAGIKDRVYSNSIYELLENGQRAGTCVLEYATPLQTLFAMSQYSQAGFSREDRLEQAKLFCRTLEDILADAPESQNNCRLIAYQEPADDSSFSLSQEVLRHLRQEEKEEVTVGSLKTSAVPSTSTMSQEPELLISGMEKPLPLRTDFS