| Assay Method Information | |
| | Ion Channel Selectivity |
| Description: | In order to address more specifically the potential selectivity issues, a counterassay was carried out for compound 2 against TRPV1 and TRPV4 ion channels, both involved in the nociception (Jhaveri M D, et al 2005. Eur. J. Neurosci. 22 (2): 361-70, Brierley S M et al, 2008, Gastroenterology. 2008 June; 134 (7):2059-69) and towards TRPA1. |
| Affinity data for this assay | |
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